TDI-11055

TDI-11055 : Inhibitor of MLLT1

Structure

Information

  • MLLT1
  • Inhibitor
  • up to 1 uM

In Vitro Validations

Uniprot ID: Q03111
Target Class: Epigenetic
Target SubClass: YEATS
Potency: Kd
Potency Value: 120 nM
Potency Assay: ITC
PDB ID for probe-target interaction (3D structure): --
Target aliases:
Protein ENL, YEATS1, LTG19, ENL, MLLT1, ENL_HUMAN, ...

DOI Reference: 10.1021/acsmedchemlett.4c00016

Uniprot ID: Q03111
Target Class: Epigenetic
Target SubClass: YEATS
Potency: IC50
Potency Value: 50 nM
Potency Assay: TR-FRET
PDB ID for probe-target interaction (3D structure): --
Target aliases:
Protein ENL, YEATS1, LTG19, ENL, MLLT1, ENL_HUMAN, ...

DOI Reference: 10.1021/acsmedchemlett.4c00016

In Cell Validations

In Vivo Data

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SERP ratings and comments


No SERP comments found for TDI-11055