STO609

ATP-competitive inhibitor of CAMKK1, CAMKK2

Structure

Information

Protein target names: CAMKK1, CAMKK2

Mechanism of action: ATP-competitive inhibitor

In Vitro Validations

Uniprot ID: Q8N5S9
Target Class: Kinase
Target SubClass: Other
Potency: Ki
Potency Value: 250 nM
Potency Assay: Autophosphorylation of CaM-KKα and -β
PDB ID for probe-target interaction (3D structure): --
Target aliases:
Calcium/calmodulin-dependent protein kinase kinase ...

DOI Reference: 10.1074/jbc.M201075200

Uniprot ID: Q8N5S9
Target Class: Kinase
Target SubClass: Other
Potency: IC 50
Potency Value: 380 nM
Potency Assay: in vitro kinase assays
PDB ID for probe-target interaction (3D structure): --
Target aliases:
Calcium/calmodulin-dependent protein kinase kinase ...

DOI Reference: 10.1074/jbc.M201075200

In Cell Validations

In Vivo Data

No in Vivo Validations

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SERP ratings and comments


SERP Ratings

In Cell Rating

(last updated: 29 Aug 2016 )

SERP Ratings

In Cell Rating

(last updated: 29 Aug 2016 )

SERP Ratings

In Cell Rating

(last updated: 29 Aug 2016 )