Prednisolone

Prednisolone : Glucocorticoid-competitive agonist of NR3C1

Structure

Information

  • NR3C1
  • Glucocorticoid competitive, Agonist

In Vitro Validations

Uniprot ID: P04150
Target Class: Nuclear Receptor
Target SubClass: Nuclear hormone receptor
Potency: Ki
Potency Value: 2.5 nM
Potency Assay: GR binding assays
PDB ID for probe-target interaction (3D structure): 6W9K 6W9K
Target aliases:
Glucocorticoid receptor, GRL, NR3C1, GCR_HUMAN, GR ...

DOI Reference: 10.1021/jm010228c

In Cell Validations

In Vivo Data

No in Vivo Validations

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SERP ratings and comments


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