Ogerin

Positive Allosteric Modulator of GPR68

Structure

SERP Rating

In Cells

(1 ratings)

In Model Organisms

(1 ratings)

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Probe Ogerin is in the process of SERP review.

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Information

Protein target names: GPR68

Mechanism of action: Positive Allosteric Modulator

Primary References:

DOI - 10.1038/nature15699

Additional Data

SGC image SGC Chemical Probe Collection

Probe Availability:

MedChemExpress
Sigma
MCULE
TOCRIS

In Vitro Validations

No in Vitro Validations

In Cell Validations

In Vivo Data

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SERP ratings and comments

SERP Ratings

In Cell Rating

In Model Organisms

SERP Comments:

Ogerin has moderate affinity at two GPCRs, 5-HT2B and the A2A receptor.

(last updated: 18 Oct 2020 )