NVP-2

Inhibitor, ATP competitive of CDK9

Structure

Information

Protein target names: CDK9

Mechanism of action: Inhibitor, ATP competitive

Recommended in-cell concentration:
250 to 1000 nM

In Vitro Validations

Uniprot ID: P50750
Target Class: Kinase
Target SubClass: CMGC
Potency: IC50
Potency Value: 0.514 nM
Potency Assay: Cdk9/CyclinT1 IMAP
PDB ID for probe-target interaction (3D structure): --
Target aliases:
Cyclin-dependent kinase 9, TAK, CDC2L4, CDK9, CDK9 ...

DOI Reference: 10.1038/nchembio.2538

In Cell Validations

In Vivo Data

No in Vivo Validations

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(last updated: 7 Jul 2021 )