MSD-M1PAM

Positive allosteric modulator of CHRM1

Probe MSD-M1PAM is in the process of SERP review.

Please continue to check back for new reviews and commentary.

Additional Data

Probe Availability:

No in Vitro Validations

Potency assay (off target): > 700-fold selectivity over CHRM2, CHRM3, CHRM4 Clean GPCR scan

Probe Selectivity in Vitro:

Closest off-targets (Panlabs): PTPN2: IC50 = 10 µM @ 10 µM;

No SERP comments found for MSD-M1PAM