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up to 10 uM
1H NMR (400MHz, CDCl3, 25 ºC) δ 1.40 (m, 6H), 3.67 (s, 2H), 4.39 (m, 6H), 6.95 (m, 3H), 7.26 (m, 2H), 7.37 (d, J = 8.4 Hz, 2H), 8.16 (d, J = 8.4 Hz, 2H), 8.45 (s, 2H)
GW1100 has no effect on the GPR120‐mediated stimulation of intracellular Ca2+ release. Outside target family: Shown to be at least 100‐fold selective against 220 other GPCRs, 60 kinases, 63 proteases, seven integrins and 20 nuclear receptors including PPARα, δ and γ, with the exception of the oxytocin receptor, for which it acted as an antagonist with a pIC50 6.9
