dBRD9

Degrader (PROTAC) of BRD9

Structure

Information

Protein target names: BRD9

Mechanism of action: Degrader (PROTAC)

Recommended in-cell concentration:
100 nM

In Vitro Validations

Uniprot ID: Q9H8M2
Target Class: Epigenetic
Target SubClass: Bromodomain
Potency: IC50
Potency Value: 104 nM
Potency Assay: AlphaScreen
PDB ID for probe-target interaction (3D structure): 5TWX
Structure-activity relationship: yes
Target aliases:
Bromodomain-containing protein 9, BRD9, BRD9_HUMAN ...

DOI Reference: 10.1002/anie.201611281

In Cell Validations

In Vivo Data

No in Vivo Validations

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