BAY-876

Inhibitor of SLC2A1

Structure

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In Cells

(2 ratings)

In Model Organisms

(2 ratings)

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Information

Protein target names: SLC2A1

Mechanism of action: Inhibitor

Recommended in-cell concentration:

up to 100 nM

Aditional Data

SGC image SGC Chemical Probe Collection

Probe Availability:

In Vitro Validations

Uniprot ID: P11166

Target Class: Transporter

Target SubClass: Solute Carrier

Potency: IC50

Potency Value: 2 nM

Potency Assay: Inhibition of glucose uptake measured by measuring ATP levels using CellTiter-Glo Luminescent Cell viability assay

PDB ID for probe-target interaction (3D structure): --

Target aliases:

Solute carrier family 2, facilitated glucose trans ...

DOI Reference: 10.1002/cmdc.201600276

In Cell Validations

In Vivo Data

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SERP Ratings

In Cell Rating

In Model Organisms

(last updated: 29 Nov 2021 )

SERP Ratings

In Cell Rating

In Model Organisms

(last updated: 3 Dec 2021 )