AP-204

AP-204 : Inhibitor of STK17B

Probe AP-204 is in the process of SERP review.

Please continue to check back for new reviews and commentary.

Uniprot ID: O94768

Target Class: Kinase

Target SubClass: CAMK

Potency: IC50

Potency Value: 130 nM

Potency Assay: Eurofins enzyme assay

PDB ID for probe-target interaction (3D structure): --

Target aliases:

Serine/threonine-protein kinase 17B, DRAK2, STK17B ...

Potency assay, off target (cells): Selective over STK17A in NanoBRET IC50 2200 nM

Potency assay (off target): DiscoverX SCANmax at 1 uM provided S10 of 0.02, total number of kinases tested 403.

No SERP comments found for AP-204