XMD17-109
Unsuitables - unsuitable to be used as a chemical probe
Structure
This is unsuitable as a chemical probe: While this
compound has been used to interrogate specific protein
targets, it is not a chemical probe and should not be used
in assays that depend on a potent and selective modulator
of the protein.
Non selective compound
While this compound is selective among the kinases, it also inhibits bromodomains. The bromodomain-binding activity is sufficient to explain all of the compound's reported biological activities.