Prednisolone

Prednisolone : Glucocorticoid-competitive agonist of NR3C1

Structure

SERP Rating

In Cells

(1 ratings)

In Model Organisms

(0 ratings)

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Probe Prednisolone is in the process of SERP review.

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Information

NR3C1

Agonist

Probe Availability:

In Vitro Validations

Uniprot ID: P04150

Target Class: Nuclear Receptor

Target SubClass: Nuclear hormone receptor

Potency: Ki

Potency Value: 2.5 nM

Potency Assay: GR binding assays

PDB ID for probe-target interaction (3D structure): 6W9K, 6W9K

Target aliases:

Glucocorticoid receptor, GRL, NR3C1, GCR_HUMAN, GR ...

DOI Reference: 10.1021/jm010228c

In Cell Validations

In Vivo Data

No in Vivo Validations

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SERP ratings and comments

SERP Ratings

In Cell Rating

SERP Comments:

No solubility data No stability data No cytotoxicity data

(last updated: 18 Jun 2024 )